VI Multidyscyplinarna Konferencja Nauki o Leku

 on-line journal

Time
 Duration
 Type
 Presenting person
 Title

May 25th, Sunday

12:00 Odjazd autokarów z Uczestnikami spod Dworca Centralnego w Warszawie. Przyjazd do Przemyśla około godz. 18:00-19:00
15:00 Rejestracja Uczestników - Rejestracja Uczestników zgodnie z zakwaterowaniem. (Informację o miejscu zakwaterowanie Uczestniczy otrzymają drogą mailową) - Przemyśl-Hotel Gromada, Krasiczyn-Hotel Zamkowy
19:00 Kolacja - Kolacja w miejscu zakwaterowania - Hotel Gromada-Przemyśl, Hotel Zamkowy-Krasiczyn

May 26th, Monday

08:30 Otwarcie Konferencji
08:45 First Session - Janusz Obukowicz, Grzegorz Grynkiewicz - Conference Room Gromada Hotel
08:45 00:30:00 Invited oral Teresa Paszkowska-Reymer The Concept of the Central Strategic Program - Innovative Medicines
09:15 00:30:00 Invited oral Jan Lubiński Genetic contribution to all cancers: implications for pharmaceutical treatment
09:45 00:30:00 Invited oral Zbigniew E. Fijałek Unusual application of X-Ray diffraction in drug control – searching for counterfeit and substandard pharmaceuticals
10:15 00:20:00 Oral Krzysztof Brzózka Focus on drug discovery – new opportunities in life science sector in Poland.
10:35 00:20:00 Oral Krystyna Gryz Registration dossier of chemical active substance
10:55 Coffee break - Gromada Hotel
11:25 First Session - Janusz Obukowicz, Grzegorz Grynkiewicz - Conference Room Gromada Hotel
11:25 00:20:00 Oral Małgorzata Jarończyk The ligand binding to the serotonin transporter
11:45 00:20:00 Oral Katarzyna A. Kaźmierska Hydrogel coatings and a local drug delivery
12:05 00:20:00 Oral Lech Kozerski Novel medium for monomer proteins structure elucidation. Human insulin structure in water/ acetonitrile solvent. Search for nonamyloidogenic conditions
12:25 00:20:00 Oral Sebastian Kmiecik Protein modeling in silico: providing new targets for a drug design
12:45 00:20:00 Oral Maria Kraj Bortezomib in multiple myeloma: treatment and retreatment. A single center experience
13:10 Lunch break - Gromada Hotel
15:00 Second Session - Marek Chmielewski, Zbigniew Fijałek - Conference Room Gromada Hotel
15:00 00:30:00 Invited oral Jan Barciszewski Human brain tumor therapy through interference RNA intervention
15:30 00:30:00 Invited oral Krzysztof L. Krzystyniak Therapeutic monoclonal antibodies in clinical and scientific data*
16:00 00:20:00 Oral Zbigniew J. Kamiński Synthesis and Screening of the Library of the Supramolecular Structures Formed by N-Lipidated Oligopeptides for Selection of Host Active as Artificial Esterase
16:20 00:20:00 Oral Wojciech Łuniewski Synthesis of selected 14C radiolabelled compounds in recent investigations of new analytical method applied in accelerated drug development (EUMAPP).
16:40 Coffee break - Gromada Hotel
17:10 Discussion Panel - Discussion leader: Aleksander P. Mazurek - Towards new therapies. Introductory remarks, Grzegorz Grynkiewicz: Microdosing - clinical trials phase 0 (FP6 project:EUMAPP) - Conference Room Gromada Hotel
18:40 Free Time
20:30 Gala Banquet - Castle Courtyard in Krasiczyn

May 27th, Tuesday

08:30 Third Session - Jan Barciszewski, Wojciech T. Markiewicz - Conference Room Gromada Hotel
08:30 00:30:00 Invited oral Marek Chmielewski Strategies of the synthesis of oxa- and carba-penams and cephams
09:00 00:30:00 Invited oral Jerzy Ostrowski Integrative genomics - an essential tool for development of molecular medicine
09:30 00:20:00 Oral Maciej Mikina New phosphonate - based strategy for the synthesis of carbocyclic nucleosides: natural Neplanocin A and its unnatural enantiomer.
09:50 00:20:00 Oral Zofia Mazerska Specific metabolism of antitumor agents with cytochrome P-450 isoenzymes
10:10 00:20:00 Oral Krzysztof Kamiński N-Phenylamino derivatives of 3-substituted pyrrolidine-2,5-diones as potential anticonvulsant agents
10:30 00:20:00 Oral Maria M. Kasprzak Cytotoxic and proapoptotic in vitro activity of two novel flavone complexes of ruthenium(II)
10:50 Coffee break - Gromada Hotel
11:20 Third Session - Jan Barciszewski, Wojciech T. Markiewicz - Conference Room Gromada Hotel
11:20 00:20:00 Oral Agata B. Maciejczyk The role of the Office for Medicinal Products, Medical Devices and Biocidal Products in pharmacovigilance activities in Poland
11:40 00:20:00 Oral Aleksandra E. Mościcka-Studzińska Electrically enhanced and controlled drug delivery through buccal mucosa
12:00 00:20:00 Oral Marek T. Konieczny Comparison of traditional and new methods of drug discovery
12:20 00:20:00 Oral Sławomir Jarosz Synthesis of higher carbon sugars. Unexpected rearrangement of higher sugar allylic alcohols
12:40 00:20:00 Oral Alicja Nowaczyk Newest triazole derivative with antifungal activity: a docking study
13:00 Lunch break - Gromada Hotel
15:00 Fourth Session - Aleksander P. Mazurek, Barbara Nawrot
15:00 00:30:00 Invited oral Sergiusz Markowicz Harnessing stem cells and dendritic cells for novel therapies
15:30 00:30:00 Invited oral Teresa M. Brodniewicz Scope and  requirements   regarding    preclinical   and human clinical trials  of a  new  medicinal product,   including  biotechnology  and biosimilar products.
16:00 Coffee break - Gromada Hotel
16:30 Discussion Panel - Discussion leader: Wiesław Szelejewski - New Technologies - Conference Room Gromada Hotel
18:00 Free Time
19:30 Picnic on the San bank (Gromada Hotel)

May 28th, Wednesday
08:30 Fifth Session - Lech Kozerski, Zofia Mazerska - Conference Room Gromada Hotel
08:30 00:30:00 Invited oral Barbara Nawrot Therapeutic applications of RNAi
09:00 00:30:00 Invited oral Witold Danikiewicz Applications of Mass Spectrometry in the Analysis of Pharmaceuticals
09:30 00:30:00 Invited oral Michał Fedoryński Phase Transfer Catalysis in pharmaceutical industry – where are we?
10:00 00:20:00 Oral Marcin Nowogródzki Polyhydroxylated decalin derivatives – stereoselective approach from simple sugars via allyltin compounds
10:20 00:20:00 Oral Agnieszka Zagórska Tricyclic theophylline derivatives with arylalkylpiperazinyl moiety as CNS agents
10:40 00:20:00 Oral Stanisław Ryng Two examples of very closely related isoxazoles exhibiting opposite immunological activities
11:00 Coffee break - Gromada Hotel
11:30 Fifth Session - Lech Kozerski, Zofia Mazerska - Conference Room Gromada Hotel
11:30 00:30:00 Invited oral Gabriel Wcisło Molecular underpinnings of the targeted therapy for cancer
12:00 00:30:00 Invited oral Tadeusz Pietrucha Overview of pharmaceutical biotechnology sector in Poland
12:30 00:20:00 Oral Piotr T. Tarnowski LC/MS/MS as a tool for profiling metabolites of active substances
12:50 00:20:00 Oral Maria Bretner Anti-glioma activity of selected CK2 protein kinase inhibitors
13:10 00:20:00 Oral Stanisław Boryczka Synthesis and antiproliferative activity in vitro of (4-substituted-2-butynylthio)quinolines
13:30 Lunch break - Gromada Hotel
15:00 Coach transport to Castle Park Complex in Krasiczyn
15:30 POSTER SESSION - Gallery of the ARP in the Royal Tower
15:30 #1 Poster Małgorzata Anyżewska The evaluation of quality of Salicis cortex raw material used in pharmaceutical preparations and its comparison with raw materials collected in natural environment
15:30 #2 Poster Ewa Augustin Metabolism of antitumor 9-amino-1-nitroacridine derivative C-1748 (Capridine-beta) in human hepatoma HepG2 cells
15:30 #3 Poster Katarzyna Badowska-Rosłonek Zolmitriptan synthesis and in-process control by HPLC methods
15:30 #4 Poster Katarzyna Badowska-Rosłonek Optimization of AR-3 synthesis
15:30 #5 Poster Andrzej J. Bojarski Searching for lead molecules as potential new CNS agents in the serotonin 5-HT6 screening assay
15:30 #6 Poster Jerzy Boryski Glycosylation reactions of natural poliphenolic compounds
15:30 #7 Poster Ryszard Bugno 2-(1-Arylsulfonylpiperidin-2-yl)ethyl derivatives as 5-HT7 receptor ligands: synthesis and their affinity for 5-HT1A/5-HT2A/5-HT7/D2 receptors
15:30 #8 Poster Ryszard Bugno SAR studies of novel 5-HT7R ligands with different spacers between aryl and amine moieties
15:30 #9 Poster Paulina Bujak The evaluation of tolterodine tartrate synthesis based on patent EP 0 325 574 B1.
15:30 #10 Poster Magdalena I. Bujalska Effect of selol on the opioids activity in vincristine induced hyperalgesia.
15:30 #11 Poster Magdalena I. Bujalska Effect of the magnesium ions on analgesic activity of opioids in vincristine induced hyperalgesia model
15:30 #12 Poster Bogdan F. Bujnicki Reactions of diastereomeric sugar derived sulfites with sterically demanding organometallics
15:30 #13 Poster Kinga Burakowska High-yielded method of synthesis of voriconazole.
15:30 #14 Poster Katarzyna Buś-Kwaśnik A high-performance liquid chromatography with electrochemical detection for the determination of olanzapine in human plasma
15:30 #15 Poster Grażyna Chłoń-Rzepa New serotonin receptors ligands in the group of 8-acylamide derivatives of 1,3-dimethyl-7-[(4-phenyl- piperazin-1-yl)-alkyl]-1H-purine-2,6-(3H,7H)-dione
15:30 #16 Poster Grażyna Chłoń-Rzepa Synthesis and serotonin receptors activity of new purine-2,6-dione derivatives with arylpiperazinylalkoxy moieties
15:30 #17 Poster Agnieszka Ciesielska Synthesis of novel pyrido[1,2-c]pyrimidine derivatives as selective ligands for 5-HT1A receptors
15:30 #18 Poster Anna Czopek Homology modeling of the 5-HT1A and 5-HT2A serotonin receptors on the novel ß2-adrenergic receptor template
15:30 #19 Poster Anna Czopek Mannich bases, 5-arylimidazolidine-2,4-dione derivatives with arylpiperazine moiety, as 5-HT1A receptor ligands with serotonin transporter affinity
15:30 #20 Poster Karolina Dąbrowska-Balcerzak Quantitation of pseudoephedrine in dosage form
15:30 #21 Poster Beata Duszyńska Flexible vs partly constrained linkers in NAN-190 and PK-13 analogs investigated as 5-HT1A/5-HT7 receptor ligands
15:30 #22 Poster Zofia Dzierżewicz Chemical characteristics of melanin from the human melanoma malignum
15:30 #23 Poster Justyna Frączyk Sulfonates of N-Triazinylammonium Salts as Highly Efficient and Environmentally Friendly Triazine-Based Coupling Reagents
15:30 #24 Poster Justyna Frączyk Rate of Binding of Host Molecules to Artificial Receptors Formed by Self-Organisation of Lipidated Oligopeptides
15:30 #25 Poster Katarzyna Gobis Synthesis and tuberculostatic activity of new N’-(6-methoxypyrazine-2-carbonyl)dithiocarbazic acid esters and their amidrazone analogs
15:30 #26 Poster Aleksandra Groman Validation of an analytical procedure – control of residual 8 solvents in a pharmaceutical substance
15:30 #27 Poster Monika K. Grudzień Molecular Properties Relevant to Bioavailability of Tioconazole  and its Derivatives
15:30 #28 Poster Łukasz Izbicki Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 2.
15:30 #29 Poster Łukasz Izbicki Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 1.
15:30 #30 Poster Jolanta Janiszewska Amphiphilic dendrimeric peptides as efficient broad spectrum antimicrobial agents
15:30 #31 Poster Magdalena Jezierska-Zięba Separation of enantiomers of Z and E 3-phenylglycidic acid t-butyl ester
15:30 #32 Poster Anna Jończyk Determination of the enantiomeric purity of epinephrine in pharmaceutical preparations
15:30 #33 Poster Barbara Kąkol Isolation and purification of (2R,3S)-3-phenylisoserine hydrochloride
15:30 #34 Poster Zbigniew J. Kamiński The New Analogues of Nitrogen Mustard With One, Two or Three 2-Chloroethylamino Fragments. Reactions with Nucleophiles
15:30 #35 Poster Anna E. Kasprzycka Fucosyl thiocarbamates, synthesis and application in glycosylation
15:30 #36 Poster Sławomir Kaźmierski Structure and Molecular Dynamics of Benzodiazacoronads in the liquid phase - study of preorganization mechanism leading to planar chirality of crystals.
15:30 #37 Poster Piotr Kiełbasiński First attempts at the enzyme-promoted hydrolysis of N-acyl phosphonoamides
15:30 #38 Poster Gabriela Kłaczkow Determination of the stereoisomers of racemic α-tocopherol in pharmaceutical products by high-performance liquid chromatography and gas chromatography
15:30 #39 Poster Marta A. Kołaczek Stereoselective synthesis of highly oxygenated derivatives decalins and cyclohexanes from monosaccharides
15:30 #40 Poster Beata Kolesińska Synthesis of Building Blocks Containing Glycosyl Moieties by Using Triazinylammonium Sulfonates
15:30 #41 Poster Beata Kolesińska Transformation of Tertiary Amines into N-Triazinylated Analogues by Treatment with Chloro-1,3,5-Triazines
15:30 #42 Poster Marek T. Konieczny Application of privileged structures in new drug discovery
15:30 #43 Poster Katarzyna Korczak The Crystal Structure of distrontium salt of 5-[bis(carboxymethyl)amino]-3-carboxymethyl-4-cyano-2-thiophenecarboxylic acid
15:30 #44 Poster Anita Kornicka Synthesis, structure and biological activity of 1-[(imidazolidin-2-yl)imino]azoles*
15:30 #45 Poster Bożenna A. Kosmacińska The determination of chromatografic purity of Pramipexole Dihydrohloride Monohydrate
15:30 #46 Poster Maria Kraj Efficacy and safety of thalidomide in the treatment of relapsed and refractory multiple myeloma
15:30 #47 Poster Hanna Kruszewska Examination of antibacterial and antifungal activity of selected non-antibiotic products
15:30 #48 Poster Małgorzata Lisowska Kuźmicz Determination of the enantiomeric purity of norepinephrine in pharmaceutical preparations
15:30 #49 Poster Wojciech Łuniewski Disubstituted indolo[2,3-b]quinoline derivatives - the cytotoxic activity in vitro against various human tumor cell lines.
15:30 #50 Poster Wojciech Łuniewski Mono substituted 5H- and 6H-indolo[2,3-b]quinoline derivatives and their ability to overcome the barrier of drug resistance.
15:30 #51 Poster Marcin Mączyński Synthesis new 1,2,4-triazoline- and 1,3,4-tiadiazole - isoxazole derivatives with immunomodulatory activities
15:30 #52 Poster Wojciech T. Markiewicz Synthesis of a Polyaminooligonucleotide Combinatorial Library and Studies of Properties of Polyaminooligonucleotides
15:30 #53 Poster Zofia Mazerska The role of hepatic cytochrome P-450 enzymes in metabolism of imidazoacridinone antitumor agent, C1311 (SymadexR): studies with the hepatic NADPH:cytochrome P450 reductase null mice
15:30 #54 Poster Krzysztof Bańkowski A novel synthesis of antineoplastic drugs docetaxel and paclitaxel
15:30 #55 Poster Magdalena Milczarek New calcipotriol analogs, their toxicity and antitumor activity in vivo in comparison to the affinity with VDR and DBP
15:30 #56 Poster Stefan Mordalski Homology modeling of metabotropic glutamate receptor 2
15:30 #57 Poster Alicja Nowaczyk The nature of the interactions of oxprenolol with polypyrrole sorbent
15:30 #58 Poster Mateusz Nowak Molecular modeling explains differences in binding affinity of new potent and selective 5-HT1A ligands: arylpiperazinylalkylthiobenzoxazole derivatives
15:30 #59 Poster Mateusz Nowak Pharmacophore model of group II metabotropic glutamate receptor modulators
15:30 #60 Poster Jolanta Obniska Synthesis and anticonvulsant activity of new N-[(4-arylpiperazin-1-yl)-methyl]- 3-phenyl-pyrrolidine-2,5-dione derivatives
15:30 #61 Poster Ryszard Ostaszewski Synthesis of novel, peptidic kinase inhibitors with cytotoxic activity
15:30 #62 Poster Maria H. Paluchowska Searching for the 5-HT7 receptor ligands in the series of new 1,2,3,4-tetrahydroisoquinolines with imide fragment
15:30 #63 Poster Maria H. Paluchowska Synthesis and molecular modeling of 1,2,3,4-tetrahydroisoquinoline-based arylsulfonamides as potential 5-HT7 receptor ligands
15:30 #64 Poster Gabriela Pastuch-Gawołek Uridine derivatives of 1-thioglycosides as analogs of glycosyltransferases natural substrates
15:30 #65 Poster Gabriela Pastuch-Gawołek Uridine derivatives of heteroaryl 1-thioglycosides: synthesis and biological activity against CSFV glycoproteins
15:30 #66 Poster Elżbieta Pieniążek Crystal structure of β-adrenergic receptor as a new template in homology modeling of GPCR. Application to serotonin 5-HT1A and 5-HT7 receptors
15:30 #67 Poster Anita Pietraszek New rosiglitazone salts
15:30 #68 Poster Elżbieta Z. Pomarnacka Syntheses of N,S-substituted 4-chloro-2-mercapto-5-methylbenzenesulfonamide derivatives with potential biological activity
15:30 #69 Poster Maria Puchalska Development of HPLC and GC methods for analysis of Zolmitriptan of pharmaceutical purity
15:30 #70 Poster Jerzy Cieplik Synthesis and biological properties 1,3,7-triaryl-5-methyl-1,2,3,4-tetrahydropirimid [ 4,5-d] pirimidine derivatives.
15:30 #71 Poster Adam Redzej Synthesis of novel, thioredoxin - thioredoxin reductase inhibitors
15:30 #72 Poster Adam Redzej Selective monoacylation of alkane-α,ω-diols using crude acetone powders of animal tissues
15:30 #73 Poster Katarzyna Romanowska Title: Sex dependent antinociceptive activity and blood pressure changes in SHR, WKY and WAG rats strains after diclophenac treatment.
15:30 #74 Poster Piotr J. Rudzki Application of confidence intervals to bioanalytical method validation
15:30 #75 Poster Aleksandra Sabiniarz Structure-activity relationships in group of 2,4-dioxo-1,2,3,4-tetrahydropyrido[2,3-d]pyrimidine derivatives
15:30 #76 Poster Katarzyna M. Sarna Determination of sibutramine and desmethylsibutramine in Chinese Herbal Medicines by HPLC-ED, HPLC-MS/MS end XPRD methods
15:30 #77 Poster Joanna Wietrzyk New amino acid derivatives of 6H-indolo[2,3-b]quinolines
15:30 #78 Poster Agata Siwek Antimicrobial properties of 3-(2-methylfuran-3-yl)- 4-substituted-Δ2-1,2,4-triazoline-5-thiones
15:30 #79 Poster Sławomir Smolik Transcriptional activity of interferon γ and two subunits of its receptor as molecular markers of myocarditis
15:30 #80 Poster Jolanta Solecka JS-1, a novel isoquinoline alkaloid with antimicrobial activity isolated from Streptomyces sp. 8812
15:30 #81 Poster Anna Stankiewicz-Kranc Proline analogue of nitrosourea as a new cytotoxic prodrug
15:30 #82 Poster Sebastian Stecko Polyhydroxylated indolizidine and pyrrolizidine alkaloids. Synthesis and bioactivity.
15:30 #83 Poster Elżbieta U. Stolarczyk Isolation, structural elucidation and characterization of impurities in latanoprost
15:30 #84 Poster Marta Świtalska The cytotoxic activity of glycosides of indolo[2,3-b]quinoline derivatives.
15:30 #85 Poster Marta Świtalska The new analogs of genistein decrease mitochondrial membrane potential and activate caspase-3
15:30 #86 Poster Elżbieta Szacoń New imidazo[1,2-a][1,3,5]triazine with potential pharmacological activity
15:30 #87 Poster Adam P. Treder Synthesis and biological properties of a new family of agmatine analogues.
15:30 #88 Poster Beata Tylińska Synthesis and cytostatic activity of new 1-substituted 6H-pyrido[4,3-b]carbazole derivatives
15:30 #89 Poster Marzena Ucherek Biological action of methyl 2-[5-oxo-3,4-di-(-2-pirydyl)-1,4,5,6-tetrahydro-1,2,4-triazine-6-ylidene)acetate
15:30 #90 Poster Marzena Ucherek Synthesis and biological activity of the product obtained in the reaction of the N3-substituted amidrazones with cis-1,2-cyclohexanedicarboxylic anhydride
15:30 #91 Poster Ilona Wandzik Interactions between glycosyltransferases and 2-deoxy glycosyl derivatives of uridine simulated by molecular docking
15:30 #92 Poster Ludmiła Węglarz The effect of inositol hexaphosphate on NFkB expression in human colon cancer cells
15:30 #93 Poster Monika Wujec New derivatives of thiosemicarbazide and 1,2,4-triazole-5-thione with potential antimicrobial activity
15:30 #94 Poster Joanna Zagrodzka HPLC as a method for analytical control of synthesis and determination of tolterodine (TD-S)
15:30 #95 Poster Paweł Zajdel Solid-phase synthesis and preliminary biological investigation of arylpiperazine library as 5-HT1A and 5-HT2A receptor ligands
15:30 #96 Poster Katarzyna Zawada Oxidation status of ALDH3A1 and antioxidant capacity correlation for human saliva.
15:30 #97 Poster Maria E. Żebrowska   “Preliminary study of silicone gel sheets containing onion (Allium cepae) extract for treatment of scars”
15:30 #98 Poster Dorota Żelaszczyk Stereoselective acetylation of racemic 1-chloro-3-(2-chloro-5-methylphenoxy)propan-2-ol
15:30 #99 Poster Dorota Żelaszczyk Preparation of enantiopure (R)-hydroxy metabolite of denbufylline catalysed by immobilized Lactobacillus kefiri
15:30 #100 Poster Paweł Żero Comparison of properties of cyclic and linear glycine derived structures and their phosphorus analogues - theoretical studies
15:30 #101 Poster Andrzej Zięba New azaphenothiazine derivatives - synthesis and antibacterial properties
16:00 Coffee break - Tower Hall in Krasiczyn Castle
16:30 POSTER SESSION - Gallery of the ARP in the Royal Tower
17:15 Violin Concert
17:45 POSTER SESSION - Gallery of the ARP in the Royal Tower
18:30 Free Time
20:00 CEREMONIAL DINNER - Restaurant in the Castle

May 29th, Thursday

05:00 Śniadanie dla Uczestników wycieczki do Lwowa
05:30 Odjazd autokarów z Uczestnikami wycieczki do Lwowa
07:00 Śniadanie dla pozostałych Uczestników
09:00 Odjazd autokaru z Uczestnikami do Warszawy
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