VI Multidyscyplinarna Konferencja Nauki o Leku

 on-line journal

No.
 Presenting person
 Title
1 Małgorzata Anyżewska The evaluation of quality of Salicis cortex raw material used in pharmaceutical preparations and its comparison with raw materials collected in natural environment
2 Ewa Augustin Metabolism of antitumor 9-amino-1-nitroacridine derivative C-1748 (Capridine-beta) in human hepatoma HepG2 cells
3 Katarzyna Badowska-Rosłonek Zolmitriptan synthesis and in-process control by HPLC methods
4 Katarzyna Badowska-Rosłonek Optimization of AR-3 synthesis
5 Andrzej J. Bojarski Searching for lead molecules as potential new CNS agents in the serotonin 5-HT6 screening assay
6 Jerzy Boryski Glycosylation reactions of natural poliphenolic compounds
7 Ryszard Bugno 2-(1-Arylsulfonylpiperidin-2-yl)ethyl derivatives as 5-HT7 receptor ligands: synthesis and their affinity for 5-HT1A/5-HT2A/5-HT7/D2 receptors
8 Ryszard Bugno SAR studies of novel 5-HT7R ligands with different spacers between aryl and amine moieties
9 Paulina Bujak The evaluation of tolterodine tartrate synthesis based on patent EP 0 325 574 B1.
10 Magdalena I. Bujalska Effect of selol on the opioids activity in vincristine induced hyperalgesia.
11 Magdalena I. Bujalska Effect of the magnesium ions on analgesic activity of opioids in vincristine induced hyperalgesia model
12 Bogdan F. Bujnicki Reactions of diastereomeric sugar derived sulfites with sterically demanding organometallics
13 Kinga Burakowska High-yielded method of synthesis of voriconazole.
14 Katarzyna Buś-Kwaśnik A high-performance liquid chromatography with electrochemical detection for the determination of olanzapine in human plasma
15 Grażyna Chłoń-Rzepa New serotonin receptors ligands in the group of 8-acylamide derivatives of 1,3-dimethyl-7-[(4-phenyl- piperazin-1-yl)-alkyl]-1H-purine-2,6-(3H,7H)-dione
16 Grażyna Chłoń-Rzepa Synthesis and serotonin receptors activity of new purine-2,6-dione derivatives with arylpiperazinylalkoxy moieties
17 Agnieszka Ciesielska Synthesis of novel pyrido[1,2-c]pyrimidine derivatives as selective ligands for 5-HT1A receptors
18 Anna Czopek Homology modeling of the 5-HT1A and 5-HT2A serotonin receptors on the novel ß2-adrenergic receptor template
19 Anna Czopek Mannich bases, 5-arylimidazolidine-2,4-dione derivatives with arylpiperazine moiety, as 5-HT1A receptor ligands with serotonin transporter affinity
20 Karolina Dąbrowska-Balcerzak Quantitation of pseudoephedrine in dosage form
21 Beata Duszyńska Flexible vs partly constrained linkers in NAN-190 and PK-13 analogs investigated as 5-HT1A/5-HT7 receptor ligands
22 Zofia Dzierżewicz Chemical characteristics of melanin from the human melanoma malignum
23 Justyna Frączyk Sulfonates of N-Triazinylammonium Salts as Highly Efficient and Environmentally Friendly Triazine-Based Coupling Reagents
24 Justyna Frączyk Rate of Binding of Host Molecules to Artificial Receptors Formed by Self-Organisation of Lipidated Oligopeptides
25 Katarzyna Gobis Synthesis and tuberculostatic activity of new N’-(6-methoxypyrazine-2-carbonyl)dithiocarbazic acid esters and their amidrazone analogs
26 Aleksandra Groman Validation of an analytical procedure – control of residual 8 solvents in a pharmaceutical substance
27 Monika K. Grudzień Molecular Properties Relevant to Bioavailability of Tioconazole  and its Derivatives
28 Łukasz Izbicki Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 2.
29 Łukasz Izbicki Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 1.
30 Jolanta Janiszewska Amphiphilic dendrimeric peptides as efficient broad spectrum antimicrobial agents
31 Magdalena Jezierska-Zięba Separation of enantiomers of Z and E 3-phenylglycidic acid t-butyl ester
32 Anna Jończyk Determination of the enantiomeric purity of epinephrine in pharmaceutical preparations
33 Barbara Kąkol Isolation and purification of (2R,3S)-3-phenylisoserine hydrochloride
34 Zbigniew J. Kamiński The New Analogues of Nitrogen Mustard With One, Two or Three 2-Chloroethylamino Fragments. Reactions with Nucleophiles
35 Anna E. Kasprzycka Fucosyl thiocarbamates, synthesis and application in glycosylation
36 Sławomir Kaźmierski Structure and Molecular Dynamics of Benzodiazacoronads in the liquid phase - study of preorganization mechanism leading to planar chirality of crystals.
37 Piotr Kiełbasiński First attempts at the enzyme-promoted hydrolysis of N-acyl phosphonoamides
38 Gabriela Kłaczkow Determination of the stereoisomers of racemic α-tocopherol in pharmaceutical products by high-performance liquid chromatography and gas chromatography
39 Marta A. Kołaczek Stereoselective synthesis of highly oxygenated derivatives decalins and cyclohexanes from monosaccharides
40 Beata Kolesińska Synthesis of Building Blocks Containing Glycosyl Moieties by Using Triazinylammonium Sulfonates
41 Beata Kolesińska Transformation of Tertiary Amines into N-Triazinylated Analogues by Treatment with Chloro-1,3,5-Triazines
42 Marek T. Konieczny Application of privileged structures in new drug discovery
43 Katarzyna Korczak The Crystal Structure of distrontium salt of 5-[bis(carboxymethyl)amino]-3-carboxymethyl-4-cyano-2-thiophenecarboxylic acid
44 Anita Kornicka Synthesis, structure and biological activity of 1-[(imidazolidin-2-yl)imino]azoles*
45 Bożenna A. Kosmacińska The determination of chromatografic purity of Pramipexole Dihydrohloride Monohydrate
46 Maria Kraj Efficacy and safety of thalidomide in the treatment of relapsed and refractory multiple myeloma
47 Hanna Kruszewska Examination of antibacterial and antifungal activity of selected non-antibiotic products
48 Małgorzata Lisowska Kuźmicz Determination of the enantiomeric purity of norepinephrine in pharmaceutical preparations
49 Wojciech Łuniewski Disubstituted indolo[2,3-b]quinoline derivatives - the cytotoxic activity in vitro against various human tumor cell lines.
50 Wojciech Łuniewski Mono substituted 5H- and 6H-indolo[2,3-b]quinoline derivatives and their ability to overcome the barrier of drug resistance.
51 Marcin Mączyński Synthesis new 1,2,4-triazoline- and 1,3,4-tiadiazole - isoxazole derivatives with immunomodulatory activities
52 Wojciech T. Markiewicz Synthesis of a Polyaminooligonucleotide Combinatorial Library and Studies of Properties of Polyaminooligonucleotides
53 Zofia Mazerska The role of hepatic cytochrome P-450 enzymes in metabolism of imidazoacridinone antitumor agent, C1311 (SymadexR): studies with the hepatic NADPH:cytochrome P450 reductase null mice
54 Krzysztof Bańkowski A novel synthesis of antineoplastic drugs docetaxel and paclitaxel
55 Magdalena Milczarek New calcipotriol analogs, their toxicity and antitumor activity in vivo in comparison to the affinity with VDR and DBP
56 Stefan Mordalski Homology modeling of metabotropic glutamate receptor 2
57 Alicja Nowaczyk The nature of the interactions of oxprenolol with polypyrrole sorbent
58 Mateusz Nowak Molecular modeling explains differences in binding affinity of new potent and selective 5-HT1A ligands: arylpiperazinylalkylthiobenzoxazole derivatives
59 Mateusz Nowak Pharmacophore model of group II metabotropic glutamate receptor modulators
60 Jolanta Obniska Synthesis and anticonvulsant activity of new N-[(4-arylpiperazin-1-yl)-methyl]- 3-phenyl-pyrrolidine-2,5-dione derivatives
61 Ryszard Ostaszewski Synthesis of novel, peptidic kinase inhibitors with cytotoxic activity
62 Maria H. Paluchowska Searching for the 5-HT7 receptor ligands in the series of new 1,2,3,4-tetrahydroisoquinolines with imide fragment
63 Maria H. Paluchowska Synthesis and molecular modeling of 1,2,3,4-tetrahydroisoquinoline-based arylsulfonamides as potential 5-HT7 receptor ligands
64 Gabriela Pastuch-Gawołek Uridine derivatives of 1-thioglycosides as analogs of glycosyltransferases natural substrates
65 Gabriela Pastuch-Gawołek Uridine derivatives of heteroaryl 1-thioglycosides: synthesis and biological activity against CSFV glycoproteins
66 Elżbieta Pieniążek Crystal structure of β-adrenergic receptor as a new template in homology modeling of GPCR. Application to serotonin 5-HT1A and 5-HT7 receptors
67 Anita Pietraszek New rosiglitazone salts
68 Elżbieta Z. Pomarnacka Syntheses of N,S-substituted 4-chloro-2-mercapto-5-methylbenzenesulfonamide derivatives with potential biological activity
69 Maria Puchalska Development of HPLC and GC methods for analysis of Zolmitriptan of pharmaceutical purity
70 Jerzy Cieplik Synthesis and biological properties 1,3,7-triaryl-5-methyl-1,2,3,4-tetrahydropirimid [ 4,5-d] pirimidine derivatives.
71 Adam Redzej Synthesis of novel, thioredoxin - thioredoxin reductase inhibitors
72 Adam Redzej Selective monoacylation of alkane-α,ω-diols using crude acetone powders of animal tissues
73 Katarzyna Romanowska Title: Sex dependent antinociceptive activity and blood pressure changes in SHR, WKY and WAG rats strains after diclophenac treatment.
74 Piotr J. Rudzki Application of confidence intervals to bioanalytical method validation
75 Aleksandra Sabiniarz Structure-activity relationships in group of 2,4-dioxo-1,2,3,4-tetrahydropyrido[2,3-d]pyrimidine derivatives
76 Katarzyna M. Sarna Determination of sibutramine and desmethylsibutramine in Chinese Herbal Medicines by HPLC-ED, HPLC-MS/MS end XPRD methods
77 Joanna Wietrzyk New amino acid derivatives of 6H-indolo[2,3-b]quinolines
78 Agata Siwek Antimicrobial properties of 3-(2-methylfuran-3-yl)- 4-substituted-Δ2-1,2,4-triazoline-5-thiones
79 Sławomir Smolik Transcriptional activity of interferon γ and two subunits of its receptor as molecular markers of myocarditis
80 Jolanta Solecka JS-1, a novel isoquinoline alkaloid with antimicrobial activity isolated from Streptomyces sp. 8812
81 Anna Stankiewicz-Kranc Proline analogue of nitrosourea as a new cytotoxic prodrug
82 Sebastian Stecko Polyhydroxylated indolizidine and pyrrolizidine alkaloids. Synthesis and bioactivity.
83 Elżbieta U. Stolarczyk Isolation, structural elucidation and characterization of impurities in latanoprost
84 Marta Świtalska The cytotoxic activity of glycosides of indolo[2,3-b]quinoline derivatives.
85 Marta Świtalska The new analogs of genistein decrease mitochondrial membrane potential and activate caspase-3
86 Elżbieta Szacoń New imidazo[1,2-a][1,3,5]triazine with potential pharmacological activity
87 Adam P. Treder Synthesis and biological properties of a new family of agmatine analogues.
88 Beata Tylińska Synthesis and cytostatic activity of new 1-substituted 6H-pyrido[4,3-b]carbazole derivatives
89 Marzena Ucherek Biological action of methyl 2-[5-oxo-3,4-di-(-2-pirydyl)-1,4,5,6-tetrahydro-1,2,4-triazine-6-ylidene)acetate
90 Marzena Ucherek Synthesis and biological activity of the product obtained in the reaction of the N3-substituted amidrazones with cis-1,2-cyclohexanedicarboxylic anhydride
91 Ilona Wandzik Interactions between glycosyltransferases and 2-deoxy glycosyl derivatives of uridine simulated by molecular docking
92 Ludmiła Węglarz The effect of inositol hexaphosphate on NFkB expression in human colon cancer cells
93 Monika Wujec New derivatives of thiosemicarbazide and 1,2,4-triazole-5-thione with potential antimicrobial activity
94 Joanna Zagrodzka HPLC as a method for analytical control of synthesis and determination of tolterodine (TD-S)
95 Paweł Zajdel Solid-phase synthesis and preliminary biological investigation of arylpiperazine library as 5-HT1A and 5-HT2A receptor ligands
96 Katarzyna Zawada Oxidation status of ALDH3A1 and antioxidant capacity correlation for human saliva.
97 Maria E. Żebrowska   “Preliminary study of silicone gel sheets containing onion (Allium cepae) extract for treatment of scars”
98 Dorota Żelaszczyk Stereoselective acetylation of racemic 1-chloro-3-(2-chloro-5-methylphenoxy)propan-2-ol
99 Dorota Żelaszczyk Preparation of enantiopure (R)-hydroxy metabolite of denbufylline catalysed by immobilized Lactobacillus kefiri
100 Paweł Żero Comparison of properties of cyclic and linear glycine derived structures and their phosphorus analogues - theoretical studies
101 Andrzej Zięba New azaphenothiazine derivatives - synthesis and antibacterial properties
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