VII Multidyscyplinarna Konferencja Nauki o Leku :: VII Multidyscyplinarna Konferencja Nauki o Leku

No.	Presenting person	Title
1	Elżbieta Anuszewska	Modified SDS micelles for amino acid separation by MEKC. Application for amino acid profiling in formulations for parental use.
2	Małgorzata Anyżewska	Determination of total hypericins in St. John's wort and herbal medicinal products
3	Ewa Augustin	Antitumor triazoloacridinone C-1305 as a potent FLT3 tyrosine kinase inhibitor in human leukemia MV4;11 cells.
4	Lilianna Becan	Synthesis and in vitro anti-hepatitis B and C virus activity of the new nucleobase analogues containing thiazolo[4,5-d]pyrimidine ring system
5	Anna Bielawska	Inhibition of DNA topoisomerases I and II by G3 PAMAM-NH₂ dendrimer - modified digoxin and proscillaridin A conjugates in a cell free system
6	Krzysztof Bielawski	The effect of a novel dinuclear platinum complex with berenil and 2-picoline ligands on growth and metabolism of human breast cancer cells
7	Joanna M. Biernat	The development of a GC method for analysis of resi- dual acetic acid, triethylamine and N,N-dimethylfor- mamide in hydrochloride salts of pharmaceutical substances
8	Joanna M. Biernat	Problems of determination of selected Class 1 residual solvents (according to ICH^*)) as process impurities of some Class 3 and 2 solvents in API by GC-HS method
9	Janusz Boratyński	Antitumor activity of carrier-methotrexate conjugates.
10	Stanisław Boryczka	New acetylenic derivatives of betulin with anticancer activity
11	Grażyna Chłoń-Rzepa	Tricyclic derivatives of theophylline as potential ligands of CNS
12	Grażyna Chłoń-Rzepa	Synthesis of long-chain arylpiperazine theophylline derivatives as potential 5-HT₇ and 5-HT₆ receptors ligands
13	Ewa Chodurek	Evaluation of proliferation and cellular death of A375 cell line in the presence of HDACs inhibitors
14	Ewelina Czerniec-Michalik	HPLC Methods for Stress Testing of ZL-S Drug Substances
15	Zbigniew Dąbrowski	Research on isolation and identification of cyclolinopeptides from waste products of the flax linseed (Linum usitatissimum L.)
16	Anna Długosz	The role of estradiol in reducing the ethanol toxicity
17	Anna Długosz	Baicalin inhibits free radicals processes caused by chromium and cisplatin.
18	Danuta Drozdowska	Carbocyclic minor groove binders – endonuclease inhibition
19	Jolanta Dyniewicz	Development of dendrimeric somatostatin analogues
20	Beata Filip-Psurska	The influence of novel analogs of vitamin D₃ on the antiproliferative activity of cisplatin or doxorubicin on human promyelocytic leukaemia cell line HL-60
22	Katarzyna Gobis	Synthesis and antifungal activity of novel S-esters and S,S'-diesters of N'-(2-hydroxybenzoyl) hydrazinecarbo- dithioic acids
23	Jerzy Goliński	Synthesis of embutramide in mild conditions
24	Aleksandra Groman	Method development and validation of an analytical procedure - control of residual 2-iodopropane in Latanoprost
25	Beata M. Gruber	The possible role of HSP60 in synergistic action of anthracyclines and sulindac in HeLa cells
26	Arkadiusz R. Gruchlik	Polyunsaturated fatty acids alter expression of genes encoding antioxidant enzymes in A549 cells exposed to doxorubicin
27	Arkadiusz R. Gruchlik	Influence of troglitazone, sodium butyrate and 5-aminosalicylic acid on the chemokine ENA-78/CXCL5 secretion in the intestinal subepithelial myofibroblasts
28	Monika K. Grudzień	Molecular properties impact on bioavailability of imidazole antifungal agents.
29	Krystyna Gryz	The Pharmacopoeia in preparation and assessment of pharmaceutical, chemical and biological documentation of medicinal products
30	Jolanta Janiszewska	Basic low molecular dendrimeric peptides designed for better membrane recognition
31	Ewa Leciejewicz-Ziemecka	The European Pharmacopoeia in the Polish Pharmacopoeia
32	Katarzyna Jelonek	The influence of paclitaxel on hydrolytic degradation process in matrices obtained from aliphatic polyesters and polyestercarbonates
33	Anna Jończyk	Direct enantiomeric resolution of tamsulosin, clinically used chiral O-phenylethanolamine derivative with α₁-blocking activity
34	Łukasz S. Kaczmarek	Optimization of BR-8 synthesis
35	Barbara Kąkol	Improvement of the Phase-Transfer Catalysis (PTC) method for synthesis of L-proline derivatives
36	Agnieszka Kalicka	Application of preparative HPLC for protected peptide purification
37	Kamil K. Kamiński	Synthesis and physicochemical properties of cationic chitosan derivative for heparin complexation
38	Krzysztof Kamiński	Synthesis and anticonvulsant activity of N-substituted 8-azaspiro[4.5]decane-7,9-diones, 3-azaspiro[5.5]unde-cane-2,4-diones and 4-ethyl-4-methylpiperidine- 2,6-diones
39	Krzysztof Kamiński	Induced Fit Homology Model of the 5-HT₆ Serotonin Receptor - Application for Virtual Screening
40	Zbigniew J. Kamiński	An approach towards efficient peptide synthesis in aqueous solution
41	Małgorzata Kapral	Evaluation of transcriptional activity of genes encoding IL-6 and its receptor in colon cancer cells treated with phytic acid
42	Małgorzata Kapral	The influence of inositol hexaphosphate on the expression of genes encoding matrix metalloproteinases 2 and 9 and their tissue inhibitors in human colon cancer cells
43	Anna E. Kasprzycka	Glycosyl O- and S- N-allyl thiocarbamates in the synthesis oligosaccharides.
44	Anna E. Kasprzycka	Regioselective protection of functional groups in the na- tural compounds.
45	Michał Kaza	HPLC determination of cefuroxime in human plasma
46	Zygmunt Kazimierczuk	Synthesis, antiprotozoal and antibacterial properties of new polyhalogenobenzimidazoles
47	Zygmunt Kazimierczuk	Synthesis and proapoptotic properties of new casein kinase II inhibitors
48	Katarzyna Kempińska	Steroid profile of Asplenium cuneifolium
49	Gabriela Kłaczkow	Determination of impurities in medical products containing metformin hydrochloride
50	Patrycja Kleczkowska	H-Dmt-D-Lys-Phe-Phe-OH, a tetrapeptide metabolite of the opioid-neurotensin hybrid peptide PK20, expresses high antinociception
51	Szymon Kłossowski	Synthesis and biological evaluation of new inhibitors of thioredoxin - thioredoxin reductase.
52	Beata Kolesińska	Synthesis and Antimicrobial Activity of P-Tria- zinylphosphonium Salts
53	Michał Koliński	Molecular dynamics of ligand binding and concurrent activation steps in opioid receptors
54	Tomasz Kosmalski	Synthesis of fluorinated 2-arylo-3-aroilbenzo[b]furanes
55	Piotr Kosson	New tachykinin-opioid chimeric analogues as potential new analgesics
56	Cezary J. Kowalski	Differences in concentrations of tramadol and its major metabolites after per os sustained release tablet or per rectum suppository application.
57	Joanna D. Kozak	Functional activity of new derivatives of dextromethorphan as allosteric inhibitors of α3β4 nicotinic acetylocholine receptor.
58	Katarzyna A. Koziak	In the quest for a new endothelium-protecting drug among escin derivatives
59	Anna D. Kozioł	An asymmetric synthesis of 4-aryloxyazetidin-2-ones and 3,4-benzo-2-hydroxycephams
60	Wojciech Cybulski	Tiamulin hydrogen fumarate - veterinary uses and HPLC method of determination in premixes and medicated feeds
61	Wojciech Cybulski	Pharmacokinetic parameters of amoxicillin in pigs and poultry
62	Hanna Kruszewska	Examination of antimicrobial activity of selected non-antibiotic products
63	Marek Kubiszewski	Determination of reaction progress in synthesis of EE-3 by NMR technique
64	Agnieszka Kuczyńska	Anti-oxidativeproperties of prenylflavonoids isolated from hops (Humulus lupulus L.)
65	Rafał J. Kurczab	Examination of 5-HT₆ receptor affinity in the group of arylsulfonamide derivatives
66	Rafał J. Kurczab	Identification of Novel 5-HT₇R Ligands via Multistep Virtual Screening of Commercially Available Compounds Databases
67	Katarzyna Kurzepa	Application of fermentation in protein hydrolysates utilisation
68	Barbara Kwiatkowska-Patzer	Spinal cord peptide epitopes ameliorate immunological reaction in experimental allergic encephalomyelitis /eae/
69	Katarzyna Jelonek	Comparison of accelerated and real-time cyclosporine A release testing from poly(L-lactide-co-trimethylene carbonate) matrices
70	Anna A. Leśniak	Assessment of analgesic potency of biphalin in a mouse model of cancer pain
71	Małgorzata Lisowska Kuźmicz	Application of carbohydrate based chiral stationary phase for resolution of fenoterol, clinically used chiral drug
72	Hanna Liszkiewicz	Synthesis and antiproliferative activity in vitro of pyridodiazepine derivatives.
73	Katarzyna Lubelska	The possible effect of sulforaphane on the bioavailability of drugs
74	Katarzyna Lubelska	Antiprolfelative and cytotoxic effect of 5-fluorouracil and sulforaphane in Chinese hamster lung fibroblast cell line
75	Wojciech Łuniewski	Opimisation of preparation of TZ-6
76	Marcin Mączyński	Research into transformations of 5-amino-3-methyl- 4-isoxazolecarboxylic acid hydrazide under orthoesters influence
77	Marcin Mączyński	Electrochemical studies of Pt (II) complexes with potential bioreductive properties
78	Marta Majewska	The development of the analytical methods for studying capsules containing Temozolomide active substance
79	Adam Mames	An entry to carbapenams via asymmetric Kinugasa reaction involving cyclic nitrones and terminal acetylenes
80	Agnieszka Markowska	Tripeptides with C-terminal arginine as potential inhibitors of urokinase
81	Magdalena Milczarek	The influence of (24R)-1,24- dihydroxyvitamin D₃ on the anticancer activity of 5-fluorouracil in human colon cancer model
82	Stefan Mordalski	Interaction fingerprints patterns. Binding mode analysis of mGlu2 receptor model based on docking studies
83	Mateusz Nowak	In vitro and in vivo evaluation of novel Pim kinase inhibitors with potent anticancer activity
84	Jolanta Obniska	Synthesis and anticonvulsant activity of new N-[4-(arylpiperazin 1-yl)]- 1,3-dioxo-1,3-dihydro-2H- isoindole- and 1,3-dioxooctahydro-2H-isoindole-2-carboxa- mides
85	Jolanta Obniska	Synthesis and anticonvulsant activity of new N-Mannich bases derived from 5-cyclopropyl-5-(4-chlorophenyl)- imidazolidine-2,4-diones
86	Zbigniew Ochal	Enzyme-catalyzed synthesis of (R)-2-(1-methyl-2-pyrro- lidine)ethanol - clemastine substrate
87	Arkadiusz Orchel	Growth of human fibroblasts in the presence of 6-hydroxyhexanoic acid
88	Elżbieta Pajtasz-Piasecka	Effect of cyclophosphamide or 5-fluorouracil-based therapy supported by cellular vaccines on induction of immunity against transplantable MC38 colon carcinoma
89	Gabriela Pastuch-Gawołek	(5-Nitro-2-pyridyl) 1-thioglycosides: application in synthesis of analogues of glycosyltransferases natural substrates
90	Gabriela Pastuch-Gawołek	Glycoconjugates, products of uridine derivatives phosphitylation and oxidation as glycosyltransferases potential inhibitors
91	Jadwiga Paszkowska	Study on lipophilicity of selected uridine derivatives
92	Edyta B. Pesta-Dynda	Development of RP HPLC method for the analysis of calcipotriol in cream and ointment
93	Anita Pietraszek	A novel synthesis of 19-nor analogs of vitamin D
94	Anita Płazińska	3D-QSAR modeling of binding affinities and functional activities for the set of β₂ adrenergic receptor agonists.
95	Anita Płazińska	Docking Study of fenoterol derivatives to the β₂ adrenergic receptor. Molecular dynamic simulations for selected agonist-β₂-AR complexes.
96	Krystyna Poręba	Catalytic synthesis and antiproliferative activity in vitro of polisubstituted isoxazolopyridine derivatives.
97	Mateusz Psurski	Could the calorically restricted ketogenic diet be an effective alternative or supportive therapy for breast cancer?
98	Mateusz Psurski	Comparison of antiproliferative activity of the natural isothiocyanates and their mercapturic derivatives.
99	Magdalena A. Radomska	Submerged cultivation of Streptomyces sp. 8812 in media containing different sources of nitrogen and carbon
100	Katarzyna Sidoryk	The synthesis of ezetimibe with high stereochemical purity
101	Katarzyna Sidoryk	New amino acid and peptide derivatives of 5H-indolo[2,3-b]quinoline and their biological activity.
102	Sylwia K. Sitek	Comparison of UPLC and HPLC using Flutamide as an example
103	Agata Siwek	Synthesis and in vitro antibacterial evaluation of 1-substituted-4-ethoxycarbonylmethylthiosemicarbazides and products of their dehydrocyclization
104	Agata Siwek	Synthesis, antimicrobial, and pharmacological properties of thiadiazole derivatives
105	Andrzej M. Składanowski	New acridine-tuftsin conjugates with cytotoxic properties and increased specificity toward tumor cells
106	Sławomir Smolik	Microsatellite markers analysis in the treatment and diagnosis of familial hypertrophic cardiomyopathy
107	Sławomir Smolik	The chelation ability of chosen metal ions by protective ointments containing Na₂H₂EDTA and aminoacid
108	Jolanta Solecka	Novel bioactive metabolites
109	Magdalena Soluch	Straightforward Methodology for the Stereoselective Synthesis of Benzo[a]- and Indolo[2,3-a]quinolizidines
110	Magdalena Soluch	A Novel Method for the Synthesis of Ezetimibe Precursor
111	Marta K. Sowińska	Dendrimeric peptides with affinity to opioid receptors - complexation properties
112	Elżbieta U. Stolarczyk	The use of the hyphenated LC-MS/MS technique for the characterisation of impurity profile of Quetiapine during drug development
113	Marta Świtalska	Analogs of genistein and its possible anti-metastatic properties
114	Elżbieta Szacoń	New 1-(2-pirydynyl)-6-substituted imidazo[1,2-a][1,3,5]- triazine with potential pharmacological activity.
115	Aleksandra M. Szczucińska	Natural compositions with antioxidative properties
116	Wiesław Szeja	Application of 2-Nitroglycals in the Synthesis of Biologically Active Glycoconjugates
117	Katarzyna Buś-Kwaśnik	LC/MS/MS determination of exemestane in human plasma
118	Katarzyna M. Targowska-Duda	Molecular modeling of allosteric modulation of nicotinic acetylcholine receptor by different classes of ligands
119	Kinga Trzcinska	Structural characterization of PX-S
120	Wiesława Walisiewicz-Niedbalska	CLA derivatives as functional food compounds
121	Jarosław Walory	CHO cell line with stable expression of the HTRA1 gene as a tool for studying functional activity of 5-HT_1A receptor ligands
122	Sławek Wicherkiewicz	The development of the spectrofotometric and HPLC method for studying enteric coated capsules containing Duloxetine Hydrochloride active substance
123	Katarzyna Wiglusz	Effects of nonenzymatic glycosylation and fatty acids presence on meloxicam binding to human serum albumin
124	Małgorzata Milczarek	Anticancer activity of new coordinative palladium (II) complexes.
125	Anna M. Wójcicka	Synthesis and antitumor activity of novel 6-phenyl-2,7-naphthyridine derivatives.
126	Joanna Zagrodzka	Analytical control of synthesis and determination of BR-S by HPLC
127	Monika Wujec	The antiviral and virucidal activity of novel 2-[(4-methyl-4H-1,2,4-triazol-3-yl) sulfanyl]acetamide derivatives
128	Joanna Zagrodzka	HPLC method as an analitycal control of synthesis and determination of TZ-S
129	Paweł Zajdel	Quinolinesulfonamides as potential 5-HT₇ and 5-HT_1A receptor ligands
130	Paweł Zajdel	A novel handle for chemistry on solid support: the Pipecolic linker
131	Jadwiga R. Zawisza-Puchałka	Antiproliferative activity of novel synthetic genistein glycoside derivatives
132	Paweł Żero	Cyclohexaglycine as a potential ionophore
133	Marta Zezula	Validation of a HPLC method for LI-S analysis
134	Anna M. Zielińska	Stability study of the coated tablets containing clopidogrel bisulfate as the active substance
135	Tomasz Giller	Iontophoretic delivery of selected antiparkinsonian agents in vitro
136	Maria Puchalska	Investigation of unknown impurity of TD-S by HPLC-MS
137	Wojciech J. Gutman	New phenylpropanoic acid derivative with antidiabetic potential acting as a partial PPAR gamma agonist – preclinical studies.
138	Witold S. Cieśliński	The new solvates of docetaxel and C₂-C₃ alkyl esters of formic acid and their use for API’s preparation.
139	Marcin Feder	Computer aided development of dual p53-Mdm2/Mdm4 inhibitors
140	Witold S. Cieśliński	Docetaxel trihydrate - polymorphous studies and the new useful method to obtaining one of polymorph.
141	Maura D. Malińska	Experimental and theoretical charge density studies on a model analogue of vitamin D

VII Multidyscyplinarna Konferencja Nauki o Leku

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